1. Signaling Pathways
  2. GPCR/G Protein
  3. Vasopressin Receptor
  4. Vasopressin Receptor Inhibitors

Vasopressin Receptor Inhibitors

V1a Receptor 

V1b Receptor 

V2 Receptor 

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Vasopressin Receptor Inhibitors, Agonists, Antagonists & Activators
Product Name V1a Receptor  V1b Receptor  V2 Receptor  Purity
Conivaptan hydrochloride    
V2 Receptor 
99.92%
Argipressin    
V2 Receptor 
99.82%
Tolvaptan    
V2 Receptor 
99.96%
Lixivaptan    
V2 Receptor 
99.30%
Fedovapagon    
V2 Receptor , EC50: 24 nM
99.14%
Vasopressin Dimer (parallel) (TFA)    
V2 Receptor 
99.55%
TC OT 39
Avprla vasopressin receptor, Ki: 300 nM
   
Vasopressin Dimer (anti-parallel) (TFA)    
V2 Receptor 
Mozavaptan-d6    
V2 Receptor 
Pecavaptan
human V1a Receptor, IC50: 3.6 nM
canine V1a Receptor, IC50: 4.4 nM
 
human V2 Receptor, IC50: 1.7 nM
canine V2 Receptor, IC50: 1.3 nM
Conivaptan    
V2 Receptor 
L-364918    
V2 Receptor , Ki: 2400 nM
Tolvaptan-d7    
V2 Receptor